Hexarelinyog hluavtawsKev loj hlob hormone secretagogue peptide (GHS)thiab muaj zogGHSR-1a agonist, tsim los txhawbendogenous loj hlob hormone (GH) tso tawm. Nws belongs rau lubghrelin mimetic tsev neegthiab yog tsim los ntawm rau cov amino acids (ib hexapeptide), muab kev txhim kho metabolic stability thiab muaj zog GH-tso tawm los piv rau cov analogs ua ntej xws li GHRP-6.
Hexarelin tau kawm dav rau nws cov ntawv thov hauvendocrinology, nqaij nkoos, kho plawv, thiab kev kho kev laus, vim nws lub peev xwm los nce GH thiabCov tshuaj insulin zoo li kev loj hlob 1 (IGF-1)theem tsis ncaj qha qhia cov tshuaj hormones sab nraud.
Hexarelin khi rau lubKev loj hlob hormone secretagogue receptor (GHSR-1a)nyob rau ntawm pituitary thiab hypothalamus, mimicking qhov kev txiav txim ntawmghrelin ua- lub cev tshaib plab thiab GH-tso cov tshuaj hormones.
Cov haujlwm tseem ceeb physiological:
Stimulates pulsatile GH tso tawm
Nce circulatingIGF-1qib
Txhawb nqacov teebmeem anabolic(muscle loj hlob, rov qab)
Txhawb nqarog metabolismthiabcell regeneration
Tej zaum nthuav tawmcardioprotectivethiabanti-apoptoticteebmeem
Tsis zoo li lwm yam GHS peptides, Hexarelin uaTsis muaj qhov nce cortisol lossis prolactin ntau, muab ib qho kev huv huv endocrine profile.
Txhawb nqalean lub cev lojkev loj hlob
Txhim khocov leeg kho thiab rov tsim dua tshiab
Kawm hauvsarcopenia, cachexia, thiab kev kho mob tom qab phais
Preclinical kev tshawb fawb qhiatxhim kho plawv ua haujlwmtom qab raug mob myocardial
Txomob plawv fibrosisthiab txhim khosab laug ventricular ejection feem
Muaj peev xwm siv hauvplawv tsis ua hauj lwmthiabplawv agingqauv
Ncelipolysisthiab txhim khoinsulin rhiab heev
Txhawb nqaanti-aging kholos ntawm GH / IGF-1 axis stimulation
Tej zaum yuav pab tswjpob txha ceev thiab kev noj qab haus huv ntawm kev sib koom tes
Purity ≥ 99%
Tsim los ntawmsolid-phase peptide synthesis (SPPS)
GMP zoo li cov qauv, tsawg endotoxin thiab hnyav residues
Flexible mov:R & D rau kev lag luam nplai