| Lub npe | Tirzepatide Txhaj Tshuaj |
| Purity | 99% |
| Qhov tshwm sim | Dawb Lyophilized Hmoov |
| Kev tswj hwm | Kev txhaj tshuaj subcutaneous |
| Loj | 10 mg, 15 mg, 20 mg, 30 mg, 60 mg |
| Dej | 3.0% |
| Cov txiaj ntsig | Kho Mob Ntshav Qab Zib, poob phaus |
Tirzepatide Lyophilized hmoov (60 mg)
Tirzepatide (LY3298176) yog thawj tus ua yeeb yam agonist thib ob uas tsom rau GIP (glucose-dependent insulinotropic polypeptide) thiab GLP-1 (glucagon-zoo li peptide-1) receptors. Nws tau txais kev pom zoo los ntawm US FDA thaum lub Tsib Hlis 2022 rau kev kho mob ntawm hom 2 mob ntshav qab zib mellitus (T2DM) ua ib qho ntxiv rau kev noj haus thiab kev tawm dag zog.
Cov khoom no yog muab los ua 60mg lyophilized (freeze-dried) sterile hmoov nyob rau hauv vials, uas yuav tsum tau reconstituted nrog bacteriostatic dej ua ntej kev tswj hwm. Piv nrog ib leeg GLP-1 receptor agonists xws li semaglutide los yog dulaglutide, tirzepatide qhia tau hais tias muaj txiaj ntsig zoo hauv kev txhim kho cov ntshav qabzib, txhim kho cov tshuaj insulin, thiab txhawb kev poob phaus. Cov txiaj ntsig no raug ntaus nqi rau nws cov kev sib koom ua ke ntawm kev ua haujlwm dual-receptor.
Cov txiaj ntsig tseem ceeb
Glycemic tswj
Kev tswj qhov hnyav
Mob plawv
Kev siv thiab siv
Hom 2 Ntshav Qab Zib
Obesity/Weight Management
Pom zoo Dosage Comparison
| Qhov taw qhia | Pib Dose | Titration Schedule | Common Dose | Cov koob tshuaj ntau tshaj | Ntau zaus |
|---|---|---|---|---|---|
| Hom 2 Ntshav Qab Zib | 2.5 mg ib lis piam | Nce txhua 4 lub lis piam (→ 5 → 7.5 → 10 → 12.5 → 15 → 20 → 30 → 45 → 60) | 10-30 mg ib lis piam | 60 mg ib lis piam | Ib zaug ib lub lim tiam |
| Kev rog / poob phaus | 2.5 mg ib lis piam | Nce raws li kev kam rau siab (2.5 → 5 → 7.5 → 10 → 12.5 → 15 → 20 → 30 → 45 → 60) | 30-60 mg ib lis piam | 60 mg ib lis piam | Ib zaug ib lub lim tiam |
Nco tseg:Xyuas kom txhua qhov koob tshuaj yav dhau los raug zam zoo ua ntej kev nce ntxiv.
Tej yam tshwm sim tsis zoo
Pharmacokinetics
Cov ntsiab lus
Tirzepatide 60 mg lyophilized hmoov sawv cev rau lwm tiam kev kho mob nce qib, ua ke nrog kev tswj glycemic muaj zog nrog kev poob phaus zoo heev thiab muaj peev xwm tiv thaiv kab mob plawv.
Nrog rau lub sij hawm titration maj mam (2.5 mg → mus txog 60 mg), nws tso cai rau kev ua kom ntev thiab yooj yim rau kev kho tus kheej. Nws txoj kev tswj hwm ib zaug ib lim piam txhim kho kev ua raws, ua rau nws yog qhov kev xaiv tshiab thiab muaj txiaj ntsig zoo rau kev tswj hwm hom 2 mob ntshav qab zib thiab rog rog hauv cov chaw kho mob siab thiab tshawb fawb.