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Suav teb Healthy Poob CAS 96829-58-2 99% Bulk API Rimonbant Cetilistat Orlistat

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CAS Nr .: 96829-58-2

Cov mis mos molecular: C29H53NO5

Molecular Luj: 495.73

EINECS Tus lej: 639-755-1

Kev sib hloov tshwj xeeb: D20-32.0 ° (c = 1inchloroform)

Kub taw tes: 615.9 ± 30.0 ° C (Predicted)

Ceev: 0.976 ± 0.06g / cm3 (Predicted)

Cia txias: 2-8 ° C

 


Product Detail

Khoom cim npe

Ua raws li kev ntseeg ntawm "Tsim cov khoom ntawm sab saum toj ntawm ntau yam thiab tsim cov phooj ywg nrog cov neeg niaj hnub no los ntawm thoob plaws lub ntiaj teb", peb ib txwm muab qhov kev txaus siab ntawm cov neeg yuav khoom nyob rau hauv thawj qhov chaw rau Quoted nqe rau Tuam Tshoj noj qab haus huv poob phaus CAS 96829-58-2 99% Bulk API Rimonbant CetilistatOrlistat, Txij li thaum tsim nyob rau hauv thaum ntxov 1990s, peb tau tam sim no tsim peb muag network nyob rau hauv teb chaws USA, lub teb chaws Yelemees, Asia, thiab ntau lub teb chaws Middle Eastern. Peb lub hom phiaj kom tau txais cov khoom lag luam zoo tshaj plaws rau thoob ntiaj teb OEM thiab tom qab muag khoom!
Ua raws li kev ntseeg ntawm "Tsim cov khoom ntawm sab saum toj ntawm ntau yam thiab tsim cov phooj ywg nrog cov neeg niaj hnub no los ntawm thoob plaws lub ntiaj teb", peb ib txwm muab kev nyiam ntawm cov neeg yuav khoom hauv thawj qhov chaw rauSuav teb 96829-58-2, Orlistat, Nrog rau lub xeev-ntawm-tus-kos duab kev lag luam tawm tswv yim zoo thiab 300 tus neeg ua haujlwm txawj ua haujlwm nyuaj, peb lub tuam txhab tau tsim txhua yam kev daws teeb meem xws li chav kawm siab, chav nruab nrab mus rau chav kawm qis. Qhov kev xaiv tag nrho ntawm cov khoom zoo no muab peb cov neeg siv khoom sib txawv xaiv. Dhau li ntawd, peb lub tuam txhab ua raws li cov khoom lag luam zoo thiab tus nqi tsim nyog, thiab peb kuj muab koj cov kev pabcuam OEM zoo rau ntau lub npe nrov.

Product Detail

Lub npe Leuprorelin
CAS nr 53714-56-0
Cov mis mos molecular C59H84N16O12
Molecular hnyav 1 209.4
EINECS Number 633-395-9
Kev sib hloov tshwj xeeb D25 -31.7 ° (c = 1 hauv 1% acetic acid)
Qhov ntom 1.44 ± 0.1 g / cm3 (Kev kwv yees)
Kev cia khoom -15 ° C
Daim ntawv Tsis zoo
Acidity coefficient (pKa) 9.82 ± 0.15 (Predicted)
Dej solubility Soluble hauv dej ntawm 1mg / ml

Synonyms

LH-RHLEUPROLIDE;LEUPROLIDE;LEUPROLIDE(HUMAN);LEUPRORELIN;[DES-GLY10,D-LEU6,PRO-NHET9]-LUTEINISINGHORMONE-RELEASINGHORMONEHUMAN;(DES-GLY10,D-LEU6,PRO -NHET9)-LUTEINIZINGHORMONE-RELEASINGHORMONE;(DES-GLY10,D-LEU6,PRO-NHET9)-LUTEINIZINGHORMONE-RELEASINGFACTOR;[DES-GLY10,D-LEU6,PRO-NHET9]-LH-RH()

Pharmacological nyhuv

Leuprolide, goserelin, triprelin, thiab nafarelin yog ntau yam tshuaj uas feem ntau siv hauv kev kho mob kom tshem tawm zes qe menyuam rau kev kho mob cancer mis premenopausal thiab mob qog noj ntshav prostate. (hu ua GnRH-ib tshuaj), GnRH-ib cov tshuaj zoo sib xws hauv cov qauv rau GnRH thiab sib tw nrog pituitary GnRH receptors. Ntawd yog, gonadotropin secreted los ntawm pituitary txo qis, uas ua rau txo qis hauv kev sib deev hormone secreted los ntawm zes qe menyuam.

Leuprolide yog ib qho gonadotropin-tso hormone (GnRH) analog, peptide muaj li ntawm 9 amino acids. Cov khoom no tuaj yeem cuam tshuam kev ua haujlwm ntawm pituitary-gonadal system, tiv thaiv proteolytic enzymes thiab affinity rau pituitary GnRH receptor muaj zog dua GnRH, thiab cov haujlwm ntawm kev txhawb kev tso tawm ntawm luteinizing hormone (LH) yog li ntawm 20 npaug ntawm GnRH. Nws kuj muaj zog inhibitory nyhuv ntawm pituitary-gonad muaj nuj nqi tshaj GnRH. Hauv thawj theem ntawm kev kho mob, follicle stimulating hormone (FSH), LH, estrogen lossis androgen tuaj yeem nce ib ntus, thiab tom qab ntawd, vim qhov txo qis ntawm cov qog pituitary, qhov tso tawm ntawm FSH, LH thiab estrogen lossis androgen yog inhibited, uas ua rau muaj kev vam khom ntawm cov tshuaj hormones poj niam txiv neej. Cov kab mob sib deev (xws li mob qog noj ntshav prostate, endometriosis, thiab lwm yam) muaj kev kho mob.

Tam sim no, acetate ntsev ntawm leuprolide feem ntau yog siv nyob rau hauv kev kho mob, vim hais tias kev ua tau zoo ntawm leuprolide acetate yog ruaj khov nyob rau hauv chav tsev kub. Cov kua yuav tsum tau muab pov tseg. Nws tuaj yeem siv rau kev kho mob castration ntawm endometriosis thiab uterine fibroids, central precocious puberty, premenopausal mis cancer thiab prostate cancer, thiab kuj rau functional uterine los ntshav uas yog contraindicated los yog ineffective rau cov pa tshuaj hormones. Nws kuj tseem siv tau los ua premedication ua ntej endometrial resection, uas muaj peev xwm sib npaug ntawm cov endometrium, txo edema, thiab txo qhov nyuaj ntawm kev phais.Sticking rau kev ntseeg ntawm "Tsim cov khoom saum toj kawg nkaus thiab tsim cov phooj ywg nrog cov neeg niaj hnub no los ntawm thoob plaws lub ntiaj teb", peb ib txwm muab qhov kev txaus siab ntawm cov neeg yuav khoom nyob rau hauv thawj qhov chaw rau Quoted nqe 6 8% CAS9-89 Healthy Bulk API Rimonbant Cetilistat Orlistat, Txij li thaum tsim nyob rau hauv thaum ntxov 1990s, peb tau tam sim no tsim peb muag network nyob rau hauv teb chaws USA, lub teb chaws Yelemees, Asia, thiab ntau lub teb chaws Middle Eastern. Peb lub hom phiaj kom tau txais cov khoom lag luam zoo tshaj plaws rau thoob ntiaj teb OEM thiab tom qab muag khoom!
Quoted nqe rauSuav teb 96829-58-2, Orlistat, Nrog rau lub xeev-ntawm-tus-kos duab kev lag luam tawm tswv yim zoo thiab 300 tus neeg ua haujlwm txawj ua haujlwm nyuaj, peb lub tuam txhab tau tsim txhua yam kev daws teeb meem xws li chav kawm siab, chav nruab nrab mus rau chav kawm qis. Qhov kev xaiv tag nrho ntawm cov khoom zoo no muab peb cov neeg siv khoom sib txawv xaiv. Dhau li ntawd, peb lub tuam txhab ua raws li cov khoom lag luam zoo thiab tus nqi tsim nyog, thiab peb kuj muab koj cov kev pabcuam OEM zoo rau ntau lub npe nrov.


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