Melanotan II
Melanotan II API
Melanotan IIyog ib qho hluavtaws cyclic heptapeptide analog ntawmα-melanocyte-stimulating hormone (α-MSH), tsim rautxhawb nqa melanogenesis, txhim khuKev tiv thaiv UV, thiab modulatekev sib deev thiab metabolic muaj nuj nqi. Nws ua raws li ib tugtsis xaiv agonistntawm melanocortin receptors, tshwj xeebMC 1 R, MC3R ua, thiabMC4R ua.
Keeb kwm kawm rau nwstanningthiabphotoprotectivecov khoom, Melanotan II kuj tau qhia cov teebmeem ntawmtxhim kho libido, qab los noj mov, thiabzog tshuav, ua rau nws muaj ntau yam kev tshawb fawb peptide nrog kev txaus siab rau dermatology, endocrinology, thiab tshuaj sib deev.
Mechanism ntawm Action
Melanotan II ua haujlwm los ntawm kev ua kom muaj ntau yam melanocortin receptors:
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MC 1 R: Txhawb nqamelanin ntau lawm→ Ua kom cov tawv nqaij pigmentation thiab tiv thaiv UV
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MC3R / MC4R: Koom nrogtswj qab los noj mov, txhim kho libido, thiablub zog homeostasis
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Hla cov ntshav-hlwb barrier, cuam tshuam rau central neurohormonal pathways
Kev Tshawb Fawb thiab Kev Siv Muaj Peev Xwm
Txawm hais tias tsis pom zoo rau kev siv kho mob, Melanotan II tau kawm dav rau cov hauv qab no:
1. Daim tawv nqaij Pigmentation & UV tiv thaiv
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Txhawb nqaeumelanin synthesis, ua rauntuj tanning
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Muabyees duab-tiv thaiv teebmeemtsis muaj hnub raug
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Muaj peev xwm txo qis kev pheej hmoo mob qog noj ntshav hauv cov neeg tawv nqaij ncaj ncees
2. Kev sib deev tsis zoo
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Qhia raunce libido thiab kev sib deev arousalnyob rau hauv ob qho tib si txiv neej thiab poj niam
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Kawm raws li kev kho muaj peev xwm rauerectile kawg (ED)ntawm MC4R ua kom
3. Kev noj qab haus huv & Kev tswj qhov hnyav
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Tsibtxo qab los noj mov thiab noj movlos ntawm kev ua ntawm txoj kev hypothalamic
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Muaj peev xwm adjunct nyob rau hauvkev tshawb fawb kev rog
API Nta (los ntawm Gentolex Group)
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purity siab ≥ 99%(HPLC & LC-MS tau lees paub)
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Synthesized ntawmsolid-phase peptide synthesis (SPPS)
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Tsawg endotoxin, tsawg residual kuab tshuaj
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Muaj nyob rau hauvR & D rau kev lag luam nplai
